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编辑: 朱劼    发布日期: 2021-02-28   来源:威廉希尔体育  
2020
序号 论文名称 来源期刊 收录情况
1 Emodin   as a novel organic photocatalyst for selective oxidation of sulfides under   mild conditions RSC   Advances SCI
2 高效液相色谱-串联质谱法测定小鼠组织中的新型抗心力衰竭化合物AF-HF001 分析试验室 CSCDC
3 Synthesis   and biological evaluation of diaryl urea derivatives as FLT3 inhibitors Bioorganic   & Medicinal Chemistry Letters SCI
4 EGFR   抑制剂 AZD3759的合成工艺改进 中国药物化学杂志 CSCDE
5 奎扎替尼的合成 中国医药工业杂志 CSCDE
6 抗肿瘤药物恩曲替尼的合成工艺优化 化学试剂 统计源期刊
7 多靶点酪氨酸激酶抑制剂Lenvatinib的合成工艺优化 化学试剂 统计源期刊
8 HS-SPME-GC-MS法同时测定沙棘酒中11种酯类香气成分 分析试验室 CSCDC
9 柱前衍生化高效液相色谱法分析氨基酸原料药中的4种还原糖类杂质 分析试验室 CSCDC

 

2019年
序号 论文名称 来源期刊 收录情况
1 Determination   of an isonicotinylhydrazide derivative, a novel positive inotropic compound,   in mouse plasma by LC–MS/MS and its application to a pharmacokinetics study Journal   of Pharmaceutical and Biomedical Analysis SCI
2 气相色谱法测定奥希替尼中溶剂残留量 沈阳药科大学学报 CSCDE
3 新型正电荷标记试剂的反应优化及应用 广州化工 统计源期刊
4 Perylenequinonoid-Catalyzed[4+1]and[4+2]Annulations   of Azoalkenes:Photocatalytic Access to   1,2,3-Thiadiazole/1,4,5,6-Tetrahydropyridazine Derivatives JOURNAL   OF ORGANIC CHEMISTRY
SCI
5 Perylenequinonoid-catalyzed   photoredox activation for the direct arylation of (het)arenes with   sunlight Organic   & Biomolecular Chemistry SCI
6 Cercosporin-bioinspired   selective photooxidation reactions under mild conditions Green   Chemistry SCI
7 Cercosporin-bioinspired   photoreductive activation of aryl halides under mild conditions Journal   of Catalysis SCI
8 Visible-light   photocatalytic aerobic oxidation of sulfides to sulfoxides with a perylene   diimide photocatalyst Organic   & Biomolecular Chemistry SCI
9 氨基糖苷类抗生素的研究进展 中国新药杂志 CSCDC
10 Discovery   and biological evaluation of novel G protein‐coupled receptor 119 agonists   for type 2 diabetes Archiv   Der Pharmazie SCI
11 Design,   synthesis and biological evaluation   of 2-(4-(methylsulfonyl)phenyl)pyridine derivatives as GPR119 agonists Chemical   Biology & Drug Design SCI
12 靶向   Trk 抗肿瘤药物 larotrectinib 的新合成方法 中国药物化学杂志 CSCDE
13 Design,   synthesis, and evaluation of a series of novel phenylpropanoic acid   derivatives agonists for the FFA1 Chemical   Biology & Drug Design SCI
14 Isoliquiritigenin‐induced   vasodilation by activating large-conductance Ca2+‐activated K+ channels in   mouse mesenteric arteries CLINICAL   AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY SCI
15 Cercosporin-photocatalyzed   sp3 (C–H) activation for the synthesis of pyrrolo[3,4-c]quinolones Organic   & Biomolecular Chemistry SCI
16 Metal-Free   Cercosporin-Photocatalyzed C-S Coupling for the Selective Synthesis of Aryl   Sulfides under Mild Conditions European   Journal of Organic Chemistry SCI

 

2018
序号 论文名称 来源期刊 收录情况
1 Synthesis   and SAR of 4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline derivatives as potent   and selective CDK4/6 inhibitors European   Journal of Medicinal Chemistry SCI
2 Cu-Catalyzed   carbamoylation versus amination of quinoline N-oxide with formamides ORGANIC   & BIOMOLECULAR CHEMISTRY SCI
3 Synthesis   and biological evaluation of novel 5,6-dihydropyrimido[4,5-f] quinazoline   derivatives as potent CDK2 inhibitors BIOORGANIC   & MEDICINAL CHEMISTRY LETTERS SCI
4 可见光催化的丙炔酸酯三氟乙基化反应合成香豆素类似物 有机化学 SCI
5 N,N-二甲基甲酰胺二烷基缩醛对含N-H 化合物的N-烷基化反应 有机化学 SCI
6 新型抗血吸虫杂环化合物UPLC⁃QTOF⁃MS分析方法的建立 中国血吸虫病防治杂志 CSCDC
7 气相色谱法同时测定大蒜精油保健品中6 种活性有机硫化物 分析试验室 CSCDC
8 -葡萄糖共转运蛋白2抑制剂的研究进展 华西药学杂志 CSCDE
9 CDKs抑制剂BMS-265246的合成研究 中国药物化学杂志 CSCDE
10 抗癌新药帕布昔利布的合成工艺改进 中国药物化学杂志 CSCDE
11 TBAI   催化氨基羰基化合物与吲哚化合物的芳香化 广州化工 统计源
12 可见光催化下三氟甲基酮的选择性合成 广州化工 统计源
13 新型抗心衰化合物的合成及稳定性研究 广州化工 统计源

 

2017
序号 论文名称 来源期刊 收录情况
1 Gold-Oxazoline   Complex-Catalyzed Cross-Dehydrogenative
    Coupling of Glycine Derivatives and Alkenes
Advanced   Synthesis and Catalysis SCI
2 Transition-Metal-Free   Trifluoromethylation of Aldehyde Derivatives with Sodium   Trifluoromethanesulfinate JOURNAL   OF ORGANIC CHEMISTRY SCI
3 Characterization   and crystal structure of a novel zearalenone hydrolase from Cladophialophora   bantiana ACTA   CRYSTALLOGRAPHICA SECTION F-STRUCTURAL BIOLOGY COMMUNICATIONS SCI
4 三氟甲基亚磺酸钠实现的三氟甲基化反应研究进展 有机化学 SCI
5 AF-HF001对正常大鼠离体心脏的正性肌力及心电作用 中国药科大学学报 CSCDC
6 2型糖尿病相关的G蛋白偶联受体激动剂的研究进展 中国新药杂志 CSCDC
7 RP-HPLC-DAD法快速测定沙棘叶中6种黄酮成分 中国药科大学学报 CSCDC
8 CDK抑制剂PHA-848125的工艺优化 中国医药工业杂志 CSCDE
9 GPR119激动药MBX-2982的合成 中国医药工业杂志 CSCDE
10 沙棘叶黄酮提取工艺的单因素研究及其品类变化 广州化工 统计源
11 GPR40激动剂药效团模型的构建及验证 计算机与应用化学 统计源
12 多指标-正交试验优化沙棘叶和沙棘籽中黄酮的提取工艺 中国药房 统计源

 

2016
序号 论文名称 来源期刊 收录情况
1 5d, a novel analogue of 3-n-butylphthalide, decreases NADPH oxidase activity through the positive regulation of CK2 after ischemia/reperfusion injury ONCOTARGET SCI
2 Oxadiazole-2-oxides may have other functional targets, in addition to SjTGR, through which they cause mortality in Schistosoma japonicum PARASITES & VECTORS SCI
3 Iron-catalyzed direct α-arylation of α-amino carbonyl compounds with indoles Organic and Biomolecular Chemistry SCI
4 Immobilizing of oxo-molybdenum complex on cross-linked copolymer and its catalytic activity for epoxidation reactions CATALYSIS COMMUNICATIONS SCI
5 Cross-talk between 5-hydroxytryptamine and substance P in the melanogensis and apoptosis of B16F10 melanoma cells EUROPEAN JOURNAL OF PHARMACOLOGY SCI
6 Interferon-gamma Attenuates 5-Hydroxytryptamine-Induced Melanogenesis in Primary Melanocyte BIOLOGICAL & PHARMACEUTICAL BULLETIN SCI
7 Interleukin 10 protects primary melanocyte by activation of Stat-3 and PI3K/Akt/NF-kappa B signaling pathways CYTOKINE SCI
8 Gene Expression Profiling of H9c2 Cells Subjected to H2O2-Induced Apoptosis with/without AF-HF001 BIOLOGICAL & PHARMACEUTICAL BULLETIN SCI
9 首个针对治疗高危神经母细胞瘤的新药dinutuximab 中国新药杂志 CSCDE
10 -葡萄糖共转运体2抑制剂研究进展 中国新药杂志 CSCDE
11 Synthesis of Aromatic Amide Derivatives and Their Biological Evaluation against Protein Tyrosine Phosphatase 1B and Scr Homology-2 Domain Containing Protein Tyrosine Phosphatase-2 有机化学 SCI
12 Cross-talk between interferon-gamma and interleukin-18 in melanogenesis Journal of Photochemistry & Photobiology, B: Biology  SCI
13 天然大蒜精油对人体的排铅作用 分析科学学报 CSCDC
14 MK-3102关键中间体的合成工艺改进 广州化工 其他
15 邻氯苯甘氨酸甲酯的绿色合成工艺研究 广州化工 其他

   

2015年
序号 论文名称 来源期刊 收录情况
1 Zebrafish as a New Model for Phenotype-based Screening of Positive Inotropic Agents CHEMICAL BIOLOGY & DRUG DESIGN SCI
2 TBAI-catalyzed synthesis of alpha-ketoamides via sp(3) C-H radical/radical cross-coupling and domino aerobic oxidation TETRAHEDRON LETTERS SCI
3 Rh(I)-catalyzed decarbonylation synthesis of carbazoles via C-N cleavage TETRAHEDRON SCI
4 Palladium-Catalyzed Heck-Type Coupling via C-N Cleavage SYNLETT SCI
5 An efficient one-pot, three-component synthesis of vinyl sulfones via iodide-catalyzed radical alkenylation TETRAHEDRON SCI
6 Palladium(II)-Catalyzed C-H Acylation with Arylglycine Derivatives SYNLETT SCI
7 王不留行提取物对H_(22)荷瘤小鼠的抗肿瘤作用研究 Journal of Chinese Medicinal Materials CSCD
8 含糖结构的抗糖尿病螺环化合物研究进展 Chinese Journal New Drugs CSCD
9 手性胺拆分法制备雷美替胺 Chinese Journal of Synthetic Chemistry CSCD
10 Synthesis of novel 3-aryl-1-oxa-2,8-diazaspiro[4.5]dec-2-ene derivatives and their biological evaluation against PTP1B Chem Biol Drug Des SCI
11 Asymmetric Catalytic Carbon-Carbon Coupling Reactions via
           Cross-Dehydrogenative Coupling Reactions
CHINESE JOURNAL OF ORGANIC CHEMISTRY SCI
12 Mo Schiff base-tungstate ionic hybrid with enhanced heterogeneouscatalytic activity for epoxidation reactions Applied Catalysis A: General EI
13 Calcitonin gene-related peptide cooperates with substance P to inhibit
           melanogenesis and induces apoptosis of B16F10 cells
cytokine SCI
14 阿普司特的合成工艺研究 广州化工 统计源
15 匹伐他汀关键手性中间体的立体选择性合成 广州化工 统计源
16 新型心肌肌球蛋白激动剂CK-1827452的合成研究 广州化工 统计源
17 GPR40 激动剂的合成 广州化工 统计源
18 浅谈以唤醒使命感为目标的本科教学 当代教育实践与教学研究 统计源
19 药物合成反应课程教学改革研究 广州化工 统计源
20 浅谈药理教学改革 广州化工 统计源
2014年
序号 论文名称 来源期刊 收录情况
1 Synthesis and biological evaluation of novel bis-aromatic amides as novel PTP1B inhibitors BIOORGANIC & MEDICINAL CHEMISTRY LETTERS SCI
2 Synthesis and In Vivo Hepatoprotective Activity of Some Novel Andrographolide Derivatives LETTERS IN DRUG DESIGN & DISCOVERY SCI
3 1H-2,3-Dihydroperimidine Derivatives: A New Class of Potent Protein Tyrosine Phosphatase 1B Inhibitors MOLECULES SCI
4 Design, Synthesis, and Biological Evaluation of Andrographolide Derivatives as Potent Hepatoprotective Agents chemical biological & drug design SCI
5 Iron-Catalyzed Oxidative Phosphonation of α-sp 3-c-H  Bonds of N-Aryl Tetrahydroisoquinolines with Air as Oxidant  CHINESE J ORG CHEM SCI
6 高效液相色谱-串联质谱法测定兔血浆中吡喹酮浓度 分析试验室 CSCD
7 金催化的吲哚对α - 氨基酮的Friedel - Crafts 烷基化反应 广州化工 其他
8 微波辅助法合成手性β - 氨基酸 广州化工 其他
2013年
序号 论文名称 来源期刊 收录情况
1 基底细胞癌新型治疗药物 vismodegib 中国新药杂志 CSCD
2 治疗心力衰竭的新策略——心肌肌球蛋白激动剂 中国新药杂志 CSCD
3 寓教于研的药物化学课程教学改革研究 广州化工 统计源
4 Synthesis and SAR studies of Praziquantel derivatives with
           activity against Schistosoma japonicum
Molecules SCI
5 1-甲基-1,2,3,4-四氢异喹啉衍生物的合成及抗日本血吸虫活性评价 有机化学 SCI
6 王不留行提取物的急性毒理学研究 广州化工 统计源
2012年
序号 论文名称 来源期刊 收录情况
1 Au(III)-catalyzed intermolecular amidation of benzylic C–H bonds Organic &Biomolecular Chemistry SCI
2 Gold-Catalyzed Direct Indolation of Tetrahydroisoquinolines Chinese Journal of Chemistry SCI
3 Bu4NAuCl4 催化的H2O2 氧化的sp3-C—H 键与sp3-C—H 键的交叉偶联反应 有机化学 SCI
4 金配合物催化的吲哚对a,b-不饱和酮的Friedel-Crafts烷基化反应 有机化学 SCI
5 金催化的C—C 偶联反应研究进展 有机化学 SCI
6 药物化学课程教学改革 药学教育 统计源
7 Synthesis and Antiviral Activity of Conformational Analogues of Leucamide A Molecules SCI
8 优化制药工程专业药理学实验内容,培养学生创新能力 广州化工 统计源
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